Synthesis and Consecutive Reactions of α-Azido Ketones:
نویسندگان
چکیده
This review paper covers the major synthetic approaches attempted towards the synthesis of α-azido ketones, as well as the synthetic applications/consecutive reactions of α-azido ketones.
منابع مشابه
[Hydroxy(tosyloxy)iodo]benzene Mediated α-Azidation of Ketones
Reaction of various ketones with [hydroxy(tosyloxy)iodo]benzene (HTIB) followed by treatment of the α-tosyloxy ketones thus generated in situ with NaN3 offers a one-pot procedure for the synthesis of α-azido ketones. The HTIB used in this conversion may also be generated in situ by using iodosobenzene in combination with p-toluenesulphonic acid.
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